Medicinal Chemistry

Medicinal Chemistry of the Peripheral Nervous System – Adrenergics and Cholinergic their Biosynthesis, Metabolism and Structure Activity Relationships

• Post author:Akul Mehta
• Post published:January 27, 2011
• Post category:All Time Favorites/Articles/Medicinal Chemistry/Notes

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Sulfonated Bathophenanthroline, TBTA and Amineriazole

Catalytic Azide-Alkyne Cycloaddition: Reactivity and Application

• Post author:pssidhu
• Post published:February 15, 2011
• Post category:Medicinal Chemistry/Organic Chemistry/Presentations

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Factor Xa Inhibitors - Rivaroxaban and Apixaban

Direct Factor Xa Inhibitors as Anticoagulants

• Post author:pssidhu
• Post published:February 15, 2011
• Post category:Medicinal Chemistry/Presentations

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Metabolism of paracetamol (acetaminophen) acetanilide and phenacetin

Metabolism of Paracetamol (Acetaminophen), Acetanilide and Phenacetin

• Post author:Sweety Mehta
• Post published:August 25, 2012
• Post category:Medicinal Chemistry/Notes/Pharmacology

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pKa scale for acidity and basicity

Henderson–Hasselbalch Equation: Derivation of pKa and pKb

• Post author:Akul Mehta
• Post published:October 22, 2012
• Post category:Analytical Chemistry/Biochemistry Notes/Chemistry/Medicinal Chemistry/Notes/Organic Chemistry/Pharmaceutics

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Thin Layer Chromatography (TLC): Principle (with Animation)

• Post author:Sweety Mehta
• Post published:November 8, 2012
• Post category:Analytical Chemistry/Animations/Chemistry/Medicinal Chemistry/Notes/Organic Chemistry

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Principle of Reversed-Phase Chromatography HPLC/UPLC (with Animation)

• Post author:Akul Mehta
• Post published:December 27, 2012
• Post category:Analytical Chemistry/Animations/Chemistry/Medicinal Chemistry/Notes/Organic Chemistry/Pharmaceutics

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CYP-450 mediated Oxidative Reactions

Metabolism of Pharmaceutical Drugs and Xenobiotics

• Post author:Sweety Mehta
• Post published:January 29, 2014
• Post category:Medicinal Chemistry/Notes/Pharmacology

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Arene oxides possible reactions

Phase I Metabolism- Oxidative Reactions- Oxidation of Aromatic compounds

• Post author:Sweety Mehta
• Post published:February 15, 2014
• Post category:Medicinal Chemistry/Notes/Pharmacology

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Applications and Examples of Henderson Hasselbalch Equation

Applications and Example Problems Using Henderson–Hasselbalch Equation

• Post author:Akul Mehta
• Post published:July 24, 2014
• Post category:Analytical Chemistry/Biochemistry Notes/Chemistry/Medicinal Chemistry/Notes/Organic Chemistry/Pharmaceutics

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Aliphatic oxidation occurs at either omega or omega-1 position

Phase I Metabolism-Oxidative Reactions-Oxidation of Aliphatic and Alicyclic Compounds

• Post author:Sweety Mehta
• Post published:September 7, 2014
• Post category:Medicinal Chemistry/Notes/Pharmacology

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